Journal of Medicinal Chemistry p. 725 - 736 (1991)
Update date:2022-07-29
Topics:
Browne, L. J.
Gude, C.
Rodriguez, H.
Steele, R. E.
A new class of potent, selective, nonsteroidal inhibitors of aromatase have been discovered.The most potent member of this series is fadrozole hydrochloride, CGS 16949 A, 4-(5,6,7,8-tetrahydroimidazo<1,5-a>pyridin-5-yl)benzonitrile monohydrochloride, 26a.
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