Inorganica Chimica Acta (2019)
Update date:2022-07-29
Topics:
Okulova
Zenin
Shutkov
Kirsanov
Kovaleva
Lesovaya
Fetisov
Milaeva
Nazarov
We present the synthesis and cytotoxic potencies of new Pt(IV) complexes with lonidamine and bexarotene ligand tethered to Pt-center via a succinate-ethylenediamine linker. The in vitro results for a series of complexes with cisplatin, dichloride(ethane-1,2-diamine)platinum(II), or oxaliplatin core indicate that the addition to the structure lonidamine or bexarotene moiety can confer activity or selectivity of Pt(IV) complexes.
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