ACS Medicinal Chemistry Letters p. 450 - 453 (2012)
Update date:2022-07-30
Topics: Synthesis Inhibitors Analogues Thiosemicarbazone Cathepsin L
Song, Jiangli
Jones, Lindsay M.
Kumar, G. D. Kishore
Conner, Elizabeth S.
Bayeh, Liela
Chavarria, Gustavo E.
Charlton-Sevcik, Amanda K.
Chen, Shen-En
Chaplin, David J.
Trawick, Mary Lynn
Pinney, Kevin G.
A series of 36 thiosemicarbazone analogues containing the thiochromanone molecular scaffold functionalized primarily at the C-6 position were prepared by chemical synthesis and evaluated as inhibitors of cathepsins L and B. The most promising inhibitors f
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