Bioorganic and Medicinal Chemistry Letters p. 4117 - 4121 (2012)
Update date:2022-07-29
Topics:
Delouvrie, Benedicte
Al-Kadhimi, Katherine
Arnould, Jean-Claude
Barry, Simon T.
Cross, Darren A.E.
Didelot, Myriam
Gavine, Paul R.
Germain, Herve
Harris, Craig S.
Hughes, Adina M.
Jude, David A.
Kendrew, Jane
Lambert-Van Der Brempt, Christine
Lohmann, Jean-Jacques
Menard, Morgan
Mortlock, Andrew A.
Pass, Martin
Rooney, Claire
Vautier, Michel
Vincent, Jennifer L.
Warin, Nicolas
Potent antagonists of the integrin α5β1, which are RGD mimetics built from tyrosine are described. This paper describes the optimization of in vitro potency obtained by variation of two parts of the molecule, the central aromatic core and the amide moiety.
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Doi:10.1016/j.tet.2012.08.031
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(2012)