
Journal of Medicinal Chemistry p. 2582 - 2591 (1992)
Update date:2022-08-03
Topics:
McElroy, Andrew B.
Clegg, Stephen P.
Deal, Martyn J.
Ewan, Georg B.
Hagan, Russell M.
et al.
Incorporation of D-Pro9 into substance P related peptides is known to enhance neurokinin NK-2 receptor agonist potency and selectivity with respect to other neurokinin receptors.We now report that replacement of D-Trp9 by D-Pro9
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