Diastereoselective fluorination at benzyl position by anodic oxidation

DOI: 10.1016/S0040-4039(00)94714-2

Source and publish data:

Tetrahedron Letters p. 3137 - 3140 (1990)

Update date:2022-09-26

Topics:

Authors:

Kabore Kabore

Chebli Chebli

Faure Faure

Laurent Laurent

Marquet Marquet

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Article abstract of DOI:10.1016/S0040-4039(00)94714-2

By anodic oxidation of benzylic derivatives 1 in Et₃N,3HF/CH₃CN, diastereoselective fluorination in the α position of the electron withdrawing group is obtained. The observed stereoselectivities are discussed in connection with the i

Full text of DOI:10.1016/S0040-4039(00)94714-2

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