A versatile approach to 2,3-disubstituted indoles through the palladium-catalysed cyclization of oalkynyltrifluoroacetanilides with vinyl triflates and aryl halides

DOI: 10.1016/S0040-4039(00)74818-0

Source and publish data:

Tetrahedron Letters p. 3915 - 3918 (1992)

Update date:2022-08-04

Topics: Cyclization Aryl Halides 2,3-Disubstituted Indoles Palladium-catalysed Vinyl Triflates

Authors:

Arcadi, Antonio

Cacchi, Sandro

Marinelli, Fabio

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Article abstract of DOI:10.1016/S0040-4039(00)74818-0

The palladium-catalysed cyclization of o-alkynyltrifluoroacetanilides with vinyl triflates and aryl halides produces 2,3-disubstituted indoles in good to high yield.

Full text of DOI:10.1016/S0040-4039(00)74818-0

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