Conformationally Restrained Analogs of Sympathomimetic Catecholamines. Synthesis, Conformational Analysis, and Adrenergic Activity of Isochroman Derivatives

DOI: 10.1021/jm00073a006

Source and publish data:

Journal of Medicinal Chemistry p. 3077 - 3086 (1993)

Update date:2022-08-04

Topics:

Authors:

Macchia, Bruno

Balsamo, Aldo

Breschi, Maria Cristina

Chiellini, Grazia

Lapucci, Annalina

et al. et al.

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1021/jm00073a006

In previous papers dealing with the study of the conformations and the biopharmalogical activity of conformationally restrained analogs of sympathomimetic catecholamines (NE and ISO), proposals were advanced for the three-dimensional molecular models A, B

Full text of DOI:10.1021/jm00073a006

Products guided by the article

Product name:(2,3-dimethoxyphenyl)oxirane

Cas No:144923-98-8

R&D Labs maybe for 144923-98-8

Li's chemicals

Contact:+86-15850770348

Address:51 OF XIANGFANGCUN ROAD, Nanjing 210002, China
Shantou Baokang Pharmaceutical Co., Ltd.

Contact:+86-754-88873487

Address:5/F B Block Huangshan Bldg Huangshan Rd Shantou
Shijiazhuang Haotian Chemical Co., Ltd.

Contact:86-311-85044374

Address:293 Donggang Road
Ji'an Hairui Natural Plant Co. Ltd.

Contact:0796-8105528

Address:Meilin industry park, Qingyuan district Ji'an City, Jiangxi Province
Weihao Chemtech (ChangZhou) Co., Ltd.(expird)

Contact:051989185693

Address:NO 217 huangshan Rd ,Changzhou

Relevant to this article

Synthesis of 3-(4-Methyl-phenyl)-2-phenyl-3,4-dihydro-2H-benzo[e][1,3,2] oxazaphosphinine and Its Chalcogenides

Doi:10.14233/ajchem.2013.13937
(2013)
Metal-Free Visible-Light-Mediated Aromatization of 1,2–Dihydronaphthalenes

Doi:10.1002/ejoc.201901410
(2020)
Cyclopropane-based conformational restriction of GABA by a stereochemical diversity-oriented strategy: Identification of an efficient lead for potent inhibitors of GABA transports

Doi:10.1016/j.bmc.2013.06.063
(2013)
A convenient synthesis of lubeluzole and its enantiomer: Evaluation as chemosensitizing agents on human ovarian adenocarcinoma and lung carcinoma cells

Doi:10.1016/j.bmcl.2013.06.077
(2013)
Carbon-Carbon Bond Formation via N-Tosyliminium Ions

Doi:10.1016/S0040-4020(01)88321-6
(1992)
A novel one-pot synthesis of 7-methoxy-2-arylthieno[3,2-b]pyridine-3-ols in domino fashion

Doi:10.1016/j.tetlet.2013.07.024
(2013)

Article Doi