Conformationally Restrained Analogs of Sympathomimetic Catecholamines. Synthesis, Conformational Analysis, and Adrenergic Activity of Isochroman Derivatives

DOI: 10.1021/jm00073a006

Source and publish data:

Journal of Medicinal Chemistry p. 3077 - 3086 (1993)

Update date:2022-08-04

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Authors:

Macchia, Bruno

Balsamo, Aldo

Breschi, Maria Cristina

Chiellini, Grazia

Lapucci, Annalina

et al. et al.

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Article abstract of DOI:10.1021/jm00073a006

In previous papers dealing with the study of the conformations and the biopharmalogical activity of conformationally restrained analogs of sympathomimetic catecholamines (NE and ISO), proposals were advanced for the three-dimensional molecular models A, B

Full text of DOI:10.1021/jm00073a006

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