Conformationally Restrained Analogs of Sympathomimetic Catecholamines. Synthesis, Conformational Analysis, and Adrenergic Activity of Isochroman Derivatives

DOI: 10.1021/jm00073a006

Source and publish data:

Journal of Medicinal Chemistry p. 3077 - 3086 (1993)

Update date:2022-08-04

Topics:

Authors:

Macchia, Bruno

Balsamo, Aldo

Breschi, Maria Cristina

Chiellini, Grazia

Lapucci, Annalina

et al. et al.

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1021/jm00073a006

In previous papers dealing with the study of the conformations and the biopharmalogical activity of conformationally restrained analogs of sympathomimetic catecholamines (NE and ISO), proposals were advanced for the three-dimensional molecular models A, B

Full text of DOI:10.1021/jm00073a006

Products guided by the article

Product name:(2,3-dimethoxyphenyl)oxirane

Cas No:144923-98-8

R&D Labs maybe for 144923-98-8

Zhejiang Quzhou Jiancheng Silicone Co., Ltd.(Shanghai Jiancheng Industial and Trade Co, Ltd)

Contact:18957018777 +86-570-3888777

Address:The company production base address： Quzhou City, Zhejiang Province high-tech industrial park Nianhua Road 37
Sichuan Mianzhu Ronghong Chemical Co.,LTd

Contact:8613981840544

Address:XINSHI INDUSTRY PARK,MIANZHU,SICHUAN,CHINA
JiangXi Keyuan Biopharma Co., LTD.

Contact:+86-563-6833666

Address:Guangde Fine Chemical Zone, Anhui Province, China
Zhejiang Chemicals Import & Export Corporation

Contact:86-571-87043088

Address:No.37,Qingchun Road,Hangzhou,China
Beijing Top Science biological technology co., LTD

Contact:+86-13439059536

Address:15-1705 jre three mile, Beijing 100000,CHINA

Relevant to this article

Synthesis of 3-(4-Methyl-phenyl)-2-phenyl-3,4-dihydro-2H-benzo[e][1,3,2] oxazaphosphinine and Its Chalcogenides

Doi:10.14233/ajchem.2013.13937
(2013)
Metal-Free Visible-Light-Mediated Aromatization of 1,2–Dihydronaphthalenes

Doi:10.1002/ejoc.201901410
(2020)
Cyclopropane-based conformational restriction of GABA by a stereochemical diversity-oriented strategy: Identification of an efficient lead for potent inhibitors of GABA transports

Doi:10.1016/j.bmc.2013.06.063
(2013)
A convenient synthesis of lubeluzole and its enantiomer: Evaluation as chemosensitizing agents on human ovarian adenocarcinoma and lung carcinoma cells

Doi:10.1016/j.bmcl.2013.06.077
(2013)
Carbon-Carbon Bond Formation via N-Tosyliminium Ions

Doi:10.1016/S0040-4020(01)88321-6
(1992)
A novel one-pot synthesis of 7-methoxy-2-arylthieno[3,2-b]pyridine-3-ols in domino fashion

Doi:10.1016/j.tetlet.2013.07.024
(2013)

Article Doi