Synthesis of constrained thiorphan analogs as inhibitors of neutral endopeptidase

DOI: 10.1016/0960-894X(96)00367-8

Source and publish data:

Bioorganic and Medicinal Chemistry Letters p. 2053 - 2058 (1996)

Update date:2022-07-29

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Authors:

Beight, Douglas W.

Mehdi, Shujaath

Koehl, Jack R.

Flynn, Gary A.

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Article abstract of DOI:10.1016/0960-894X(96)00367-8

Constrained derivatives of thiorphan were prepared and found to be potent inhibitors of neutral endopeptidase 24.11.

Full text of DOI:10.1016/0960-894X(96)00367-8

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