Synthesis in dry media coupled with microwave irradiation: Application to the preparation of β-aminoesters and β-lactams via silyl ketene acetals and aldimines

DOI: 10.1016/S0040-4039(00)60361-1

Source and publish data:

Tetrahedron Letters p. 2123 - 2126 (1993)

Update date:2022-09-26

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Authors:

Texier-Boullet, Francoise

Latouche, Regine

Hamelin, Jack

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Article abstract of DOI:10.1016/S0040-4039(00)60361-1

According to the reaction conditions, silyl ketene acetals react with aldimines to give β-aminoesters (montmorillonite clay K₁₀, or para-toluenesulfonic acid) or β-lactams (KF/18 crown-6) in a few minutes under microwave irradiation.

Full text of DOI:10.1016/S0040-4039(00)60361-1

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