Analogues of capsaicin with agonist activity as novel analgesic agents; structure-activity studies. 2. The amide bond 'B-region'

DOI: 10.1021/jm00068a016

Source and publish data:

Journal of Medicinal Chemistry p. 2373 - 2380 (1993)

Update date:2022-07-30

Topics:

Authors:

Walpole Walpole

Wrigglesworth

Bevan Bevan

Campbell

Dray Dray

James James

Masdin Masdin

Perkins Perkins

Winter Winter

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Article abstract of DOI:10.1021/jm00068a016

A series of compounds incorporating replacements for the amide bond 'B- region' moiety of capsaicin have been synthesized, including vanillylamides and esters, homovanillic acid amides and esters, ureas, and thioureas. These have been tested in an in vitr

Full text of DOI:10.1021/jm00068a016

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