Analogues of capsaicin with agonist activity as novel analgesic agents; structure-activity studies. 2. The amide bond 'B-region'

DOI: 10.1021/jm00068a016

Source and publish data:

Journal of Medicinal Chemistry p. 2373 - 2380 (1993)

Update date:2022-07-30

Topics:

Authors:

Walpole Walpole

Wrigglesworth

Bevan Bevan

Campbell

Dray Dray

James James

Masdin Masdin

Perkins Perkins

Winter Winter

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1021/jm00068a016

A series of compounds incorporating replacements for the amide bond 'B- region' moiety of capsaicin have been synthesized, including vanillylamides and esters, homovanillic acid amides and esters, ureas, and thioureas. These have been tested in an in vitr

Full text of DOI:10.1021/jm00068a016

Products guided by the article

Product name:N-cyano-N'-octyl-O-phenylisourea

Cas No:150059-13-5

R&D Labs maybe for 150059-13-5

ANHUI WEICHI CHEMICAL CO.,LTD

website:http://www.weichichem.com

Contact:+8613912949432

Address:Fine Chemical Industrial Base,Wujiang town,He County,Anhui China.
waho int'l company

Contact:+86-579-85206992

Address:No 451 chouzhou north road ,room 1106 int'l business center , yiwu ,china
Xinji City Taida Sinopec Co., Ltd.

Contact:0086-311-85341278

Address:No.6, Nanhua Road,Xinji City Road,Hebei Province,China
shanghai payne pharm co.,ltd.

Contact:+86-021-58123769

Address:No.780 of Cailun Road,Zhangjiang Hi-tech Park,Pudong,Shanghai
Taizhou YOJOY Chemical Co., Ltd.

Contact:13857143241

Address:Yangfu Industrial Park, Xianju, Zhejiang, P. R. China

Relevant to this article

Microwave-assisted C-N and C-S bond-forming reactions: An efficient three-component domino sequence for the synthesis of sulfoether-decorated imidazo[1,2-A]pyridines

Doi:10.1039/c5ra05377c
(2015)
Synthesis of A-seco derivatives of betulinic acid with cytotoxic activity

Doi:10.1021/np049938m
(2004)
O-Allyl Protection of Guanine and Thymine Residues in Oligodeoxyribonucleotides

Doi:10.1021/jo00072a050
(1993)
Decomposition of 2-dialkylaminobenzoyl azides to yield isocyanates and 1,1 -dialky lindazol-1-ium-3-olates

Doi:10.1039/p19960000271
(1996)
Doi:10.1007/BF02682452
(1978)
Practical, Large-Scale Preparation of Benzoxepines and Coumarins through Rhodium(III)-Catalyzed C-H Activation/Annulation Reactions

Doi:10.1021/acs.oprd.9b00191
(2019)

Article Doi