Stereoselective Epoxidation of Phe-Gly and Phe-Phe Vinyl Isosteres

DOI: 10.1021/jo00084a037

Source and publish data:

Journal of Organic Chemistry p. 1139 - 1148 (1994)

Update date:2022-07-30

Topics:

Authors:

Jenmalm, Annika

Berts, Wei

Li, Yi-Lin

Luthman, Kristina

Csoeregh, Ingeborg

Hacksell, Uli

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Article abstract of DOI:10.1021/jo00084a037

Novel Phe-Gly and Phe-Phe isosteres have been synthesized.Vinylic isosteres of Phe-Gly and Phe-Phe were prepared by facile Julia reactions, and the resulting stereoisomers were isolated and epoxidized (m-chloroperbenzoic acid).Observed stereoselectivities

Full text of DOI:10.1021/jo00084a037

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