Synthesis and biological activity of a 1α,25-dihydroxyvitamin D2 analog bearing an amide group in the side-chain

DOI: 10.1248/cpb.45.185

Source and publish data:

Chemical and Pharmaceutical Bulletin p. 185 - 188 (1997)

Update date:2022-08-03

Topics:

Authors:

Konno, Katsuhiro

Ojima, Katsuji

Hayashi, Takaaki

Tanabe, Miyuki

Takayama, Hiroaki

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Article abstract of DOI:10.1248/cpb.45.185

Synthesis of a 1α,25-dihydroxyvitamin D₂ analog (3), in which the double bond in the side-chain is replaced by an amide group, is described. Condensation of a carboxylic acid (8) with an amine (6) gave an amide (9), which in turn led to 3 via s

Full text of DOI:10.1248/cpb.45.185

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