Synthesis of 5-methanesulfonamido-6-(2,4-difluorophenylthio)-1-indanone

Article abstract of DOI:10.1080/00397919508011826

The ethylene ketal of 5-nitro-6-bromo-1-indanone 6 was prepared via oxidation of N-(6-Bromo-5-indanyl)-acetamide 1. A subsequent mild displacement and elaboration to 6-thiosubstituted-5-amino indanone derivative 10 is also described.

Full text of DOI:10.1080/00397919508011826

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Synthetic Communications: An
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Synthesis of 5-
Methanesulfonamido-6-(2,4-
Difluorophenylthio)-1-Indanone
John Scheigetz a , Robert Zamboni a & Bruno Roy a
a Merck Frosst Centre for Therapeutic Research ,
P.O. Box 1005 Pointe Claire - Dorval, Quebec,
Canada , H9R 4P8
Published online: 16 Feb 2007.
To cite this article: John Scheigetz , Robert Zamboni & Bruno Roy (1995) Synthesis
of 5-Methanesulfonamido-6-(2,4-Difluorophenylthio)-1-Indanone, Synthetic
Communications: An International Journal for Rapid Communication of Synthetic
Organic Chemistry, 25:18, 2791-2806, DOI: 10.1080/00397919508011826
To link to this article: http://dx.doi.org/10.1080/00397919508011826
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