Journal of the Chemical Society. Perkin transactions I p. 157 - 166 (1996)
Update date:2022-09-26
Topics:
Atkinson, Robert S.
Coogan, Michael P.
Cornell, Clive L.
Oxidation of 3-amino-2-trifluoromethylquinazolin-4(3H)-one 6 with lead tetraacetate in dichloromethane gives the title 3-acetoxyamino derivative 7 which is isolable at room temperature and considerably more stable than the corresponding 2-alkyl substituted analogues. Compound 7 aziridinates alkenes in yields which are consistently higher than those from the 2-alkyl substituted analogues. Aziridinations using 3-acetoxyaminoquinazolinones bearing other electron-withdrawing groups on the 2-position of the quinazolinone ring have been examined.
View MoreContact:+86-22-26358246
Address:601-4-20, Fujiayuan, Tiantai Road, Hebei District, Tianjin, China
SHAANXI TOP PHARM CHEMICAL CO.LTD
Contact:+86-029-85733403
Address:No.108 ,west sector,south er huan,xi'an,china
Contact:+1-284-4950244
Address:Box 3069, Road Town, Tortola, British Virgin Islands
Qingzhou Baibang import and export co.,Ltd
Contact:+86-536-3265899
Address:No.338, Tuoshan Road
Wuxi Innopal International Trade CO.,LTD
Contact:+86-510-80711901-8003
Address:Room 402,Building 5,Longze Garden,No.17,South huanjiu Road,Yixing City, Jiangsu,China
Doi:10.1016/0040-4020(96)00159-7
(1996)Doi:10.1139/v67-385
(1967)Doi:10.1021/ja01520a046
(1959)Doi:10.1248/cpb.44.1647
(1996)Doi:10.1002/chem.201805082
(2019)Doi:10.1134/S1070363220060067
()
