A non-peptide ligand for the somatostatin receptor having a benzodiazepinone structure

DOI: 10.1016/0960-894X(96)00003-0

Source and publish data:

Bioorganic and Medicinal Chemistry Letters p. 267 - 272 (1996)

Update date:2022-07-29

Topics:

Authors:

Papageorgiou, Christos

Borer, Xaver

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Article abstract of DOI:10.1016/0960-894X(96)00003-0

The 1,3,4-trisubstituted-l,4-benzodiazepin-2-one 2 is a non-peptide mimic of somatostatin 1. It displaces the radioligand [¹²⁵I-Tyr³]-octreotide with an IC₅₀ of 7 μM. Copyright

Full text of DOI:10.1016/0960-894X(96)00003-0

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