Synthesis of a potent inhibitor of β-glucuronidase

DOI: 10.1016/0040-4039(96)00422-4

Source and publish data:

Tetrahedron Letters p. 2707 - 2708 (1996)

Update date:2022-08-04

Topics:

Authors:

Igarashi, Yasuhiro

Ichikawa, Mie

Ichikawa, Yoshitaka

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1016/0040-4039(96)00422-4

A new glucuronic acid-type iminosugar in which a nitrogen atom is placed in the anomeric positon was synthesized and was proven to potently inhibit β-glucuronidase, with Ki = 79 nM.

Full text of DOI:10.1016/0040-4039(96)00422-4

Products guided by the article

Product name:Acetic acid (3S,4R,5R)-4-acetoxy-5-azidomethyl-2-(4-methoxy-phenoxy)-tetrahydro-furan-3-yl ester

Cas No:177420-24-5

R&D Labs maybe for 177420-24-5

FOSHAN NANHAI ZHONGNAN PHARMACEUTICAL FACTORY

Contact:0086-0757-85609331

Address:XIAHENGTIAN INDUSTRIAL ZONE,SHAYONG VILLAGE,LISHUI TOWN
Shanghai KFSL Pharmaceutical Technology Co.,Ltd.

Contact:+86-21-39971718

Address:859 jiadingchengliu shanghai
Xian Changyue Biological Technology Co., Ltd.

website:https://www.xachangyue.com/

Contact:+86-029-88211911

Address:Keji Road NO.70
Yantai Derun Liquid Crystal Materials Co. Ltd.

website:http://www.ytderun.com

Contact:86-535-6300169

Address:ROOM 90, XIANGFU STREET, FUSHAN NEW-HIGH-TECH IDUSTRY ZONE, YANTAI
Suzhou JMS Chemical Co., Ltd.

Contact:+86-15995924277

Address:WuZhongOu suzhou new south road 89

Relevant to this article

Metalloporphyrin Cr(TPP)Cl-catalyzed Claisen rearrangement of simple aliphatic allyl vinyl ethers and its unique stereoselectivity

Doi:10.1016/j.tetlet.2005.02.136
(2005)
Synthesis of 3-(alkylthio and phenylthio)-1,1,1-trifluoroalkan-2-ones via ring opening of epoxy ethers

Doi:10.1055/s-1996-4235
(1996)
Electroluminescent nematic polymer networks with polarised emission

Doi:10.1080/10587250108025021
(2001)
Regio- and enantioselective substitution of acyclic allylic sulfoximines with butylcopper in the presence of lithium iodide and boron trifluoride

Doi:10.1021/jo960027u
(1996)
Bis(boryl)metallocenes. 1. 1,1′-bis(diisopropylboryl)cobaltocenium cation: A novel anion-binding ligand

Doi:10.1021/om960237x
(1996)
Stereoselective conjugate addition of carbon nucleophiles to chiral (E)-nitroalkenes bearing a γ-stereocenter. Origins of the observed anti selectivity

Doi:10.1016/0040-4039(96)00468-6
(1996)

Article Doi