Synthesis of unlabelled, 3H- and 125I-labelled β-CIT and its ω- fluoroalkyl analogues β-CIT-FE and β-CIT-FP, including synthesis of precursors

DOI: 10.1002/(SICI)1099-1344(199607)38:7<675::AID-JLCR880>3.0.CO;2-L

Source and publish data:

Journal of labelled compounds and radiopharmaceuticals p. 675 - 685 (1996)

Update date:2022-07-30

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Authors:

Swahn, Carl-Gunnar

Halldin, Christer

Guenther, Ilonka

Patt, Joerg

Ametamey, Simon

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Article abstract of DOI:10.1002/(SICI)1099-1344(199607)38:7<675::AID-JLCR880>3.0.CO;2-L

The full synthesis of the cocaine congener 2β-carbomethoxy-3β-(4- iodophenyl)tropane (β-CIT) and its N-fluoroalkyl analogues, fluoroethyl- and fluoropropyl-nor-β-CIT (β-CIT-FE and β-CIT-FP) starting from cocaine is described. The synthetic routes include

Full text of DOI:10.1002/(SICI)1099-1344(199607)38:7<675::AID-JLCR880>3.0.CO;2-L

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