Inverse electron demand Diels-Alder reactions of indole V. Reactions of 3-substituted indoles with heteroaromatic azadienes

DOI: 10.1016/0040-4039(96)01017-9

Source and publish data:

Tetrahedron Letters p. 5061 - 5064 (1996)

Update date:2022-08-03

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Authors:

Benson, Scott C.

Lee, Lily

Snyder, John K.

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Article abstract of DOI:10.1016/0040-4039(96)01017-9

The inverse electron demand Diels-Alder reactions of 3-substituted indoles with 1,2,4-triazines and 1,2,4,5-tetrazines proceeded in excellent yields both inter- and intramolecularly. The cycloaddition of tryptophan with a tethered 1,2,4-triazine produced a diastereomerically pure cycloadduct.

Full text of DOI:10.1016/0040-4039(96)01017-9

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