Irrevesible enzyme inhibitors. CLI. Active-site-directed irreversible inhibitors of dihydrofolic reductase derived from 5-(p-aminophenylbutyl)-2,4-diaminopyrimidines with a terminal sulfonyl fluoride.

DOI: 10.1021/jm00302a007

Source and publish data:

Journal of medicinal chemistry p. 224 - 227 (1969)

Update date:2022-09-26

Topics:

Authors:

Baker Baker

Meyer Jr.

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