Bioorganic and Medicinal Chemistry Letters p. 945 - 950 (1996)
Update date:2022-08-05
Topics:
Wang, Binghe
Zhang, Huijuan
Wang, Wei
By using model amines, several amides of coumarinic acid with the phenolic hydroxyl group protected as an ester were prepared. These model amides underwent a facile (t( 1/2 ) 1.5-31 min) lactonization to release the original amine compounds upon esterase catalyzed hydrolysis of the phenolic ester. Such a system can be used for the preparation of esterase-sensitive prodrugs of amine-containing compounds or peptids.
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