Synthesis of new 7-membered α-phenylthio cyclic oxamides: HIV inhibitors

DOI: 10.1016/S0040-4039(98)00680-7

Source and publish data:

Tetrahedron Letters p. 4021 - 4024 (1998)

Update date:2022-09-26

Topics:

Authors:

Medou Medou

Priem Priem

Quelever

Camplo Camplo

Kraus Kraus

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Article abstract of DOI:10.1016/S0040-4039(98)00680-7

Based on the concept of bioisosterism, we report the computer design and the synthesis of original 7-membered α-phenylthio cyclic oxamides with potent anti HIV-1 properties.

Full text of DOI:10.1016/S0040-4039(98)00680-7

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