Synthesis of new 7-membered α-phenylthio cyclic oxamides: HIV inhibitors

DOI: 10.1016/S0040-4039(98)00680-7

Source and publish data:

Tetrahedron Letters p. 4021 - 4024 (1998)

Update date:2022-09-26

Topics:

Authors:

Medou Medou

Priem Priem

Quelever

Camplo Camplo

Kraus Kraus

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1016/S0040-4039(98)00680-7

Based on the concept of bioisosterism, we report the computer design and the synthesis of original 7-membered α-phenylthio cyclic oxamides with potent anti HIV-1 properties.

Full text of DOI:10.1016/S0040-4039(98)00680-7

Products guided by the article

Product name:1,4-Dibenzyl-6-hydroxy-[1,4]diazepane-2,3-dione

Cas No:209522-90-7

R&D Labs maybe for 209522-90-7

jiangsu senxuan pharmaceutical and chemical co.,ltd

Contact:86-523-87982810

Address:hongqiao industrial zone,taixing,jiangsu china
Arshine Pharmaceutical Co., Limited

website:http://www.cnarshine.com

Contact:0731-88503671

Address:Room 1109.Block C3, Lugu Enterprise Plaza,No.27 Wenxuan Road,Changsha National Hi-Tech Industrial Development Zone,Hunan ,P.R.China
SHANXI XINTIANYUAN PHARMACEUTICAL CO., LTD.

website:http://www.tychemical.com

Contact:0086-358-3521713 3521715

Address:No. 1 Yintong Road, Shanxi Jiaocheng Economic Development Zone, Xiajiaying Town, Jiaocheng County, Lvliang City, Shanxi Province, China
Engineering Research Center of Pesticide, Heilongjiang Province

Contact:+86-451-86609001

Address:No.74 of Xuefu Road, Nangang District,
Jinhua City Mingzhu Pharmaceutical Co.,Ltd.

Contact:15857995878 0579-82207761

Address:No.169 Shenze Road, New Area,Jinpan Development Zone, Jinhua

Relevant to this article

Structure-activity relationships and molecular modeling of 3,5-diacyl- 2,4-dialkylpyridine derivatives as selective A₃ adenosine receptor antagonists

Doi:10.1021/jm980093j
(1998)
A trinuclear molybdenum cluster coordinated by o-nitrobenzoate

Doi:10.1107/S010827019800482X
(1998)
Syntheses, Structures, and Reactivity of Polynuclear Pyrazolato Copper(I) Complexes, Including an ab-Initio XRPD Study of [Cu(dmnpz)]₃ (Hdmnpz = 3,5-Dimethyl-4-nitropyrazole)

Doi:10.1021/ic970875n
(1998)
General solid-phase synthesis approach to prepare mechanism-based aspartyl protease inhibitor libraries. Identification of potent cathepsin D inhibitors

Doi:10.1021/ja981812m
(1998)
Heteroarylmethoxyphenylalkoxyiminoalkylcarboxylic acids as leukotriene biosynthesis inhibitors

Doi:10.1021/jm9904102
(2000)
Dynamic switching between binding sites in the complexation of macrocyclic 'push-pull' chromophores to lanthanides

Doi:10.1016/j.tet.2009.10.024
(2009)

Article Doi