Optically active antifungal azoles. X. Synthesis and antifungal activity of N-[4-(azolyl)phenyl]- and N-[4-(azolylmethyl)phenyl]-N′-[(1R,2R)-2-(2,4-difluorophenyl)-2-hydroxy -1-methyl-3-(1H-1,2,4-triazol-1-yl)propyl]-azolones

DOI: 10.1248/cpb.48.1935

Source and publish data:

Chemical and Pharmaceutical Bulletin p. 1935 - 1946 (2000)

Update date:2022-07-29

Topics:

Authors:

Kitazaki, Tomoyuki

Ichikawa, Takashi

Tasaka, Akihiro

Hosono, Hiroshi

Matsushita, Yoshihiro

Hayashi, Ryogo

Okonogi, Kenji

Itoh, Katsumi

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Article abstract of DOI:10.1248/cpb.48.1935

New optically active antifungal azoles, N-[4-(azolyl)phenyl]- and N-[4-(azolylmethyl)phenyl]-N′-[(1R,2R)-2-(2,4-difluorophenyl)-2-hydroxy -1-methyl-3-(1H-1,2,4-triazol-1-yl)propyl]azolones (1, 2, 3), were prepared in a stereocontrolled manner. Compounds 1

Full text of DOI:10.1248/cpb.48.1935

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