Bioorganic and Medicinal Chemistry Letters p. 3023 - 3026 (1999)
Update date:2022-07-31
Topics:
Couture
Gouverneur
Mioskowski
Efaroxan was synthetised by cyclisation of the tertiary alcohol 2 which was prepared by the ring opening of the gem-disubstituted epoxide 3 with ortho-metallated fluorobenzene.
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