A new approach to the synthesis of efaroxan

DOI: 10.1016/S0960-894X(99)00530-2

Source and publish data:

Bioorganic and Medicinal Chemistry Letters p. 3023 - 3026 (1999)

Update date:2022-07-31

Topics:

Authors:

Couture Couture

Gouverneur

Mioskowski

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Article abstract of DOI:10.1016/S0960-894X(99)00530-2

Efaroxan was synthetised by cyclisation of the tertiary alcohol 2 which was prepared by the ring opening of the gem-disubstituted epoxide 3 with ortho-metallated fluorobenzene.

Full text of DOI:10.1016/S0960-894X(99)00530-2

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