A new approach to the synthesis of efaroxan

DOI: 10.1016/S0960-894X(99)00530-2

Source and publish data:

Bioorganic and Medicinal Chemistry Letters p. 3023 - 3026 (1999)

Update date:2022-07-31

Topics:

Authors:

Couture Couture

Gouverneur

Mioskowski

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1016/S0960-894X(99)00530-2

Efaroxan was synthetised by cyclisation of the tertiary alcohol 2 which was prepared by the ring opening of the gem-disubstituted epoxide 3 with ortho-metallated fluorobenzene.

Full text of DOI:10.1016/S0960-894X(99)00530-2

Products guided by the article

Product name:2-benzyloxymethyl-2-ethyl-2,3-dihydro-benzofuran

Cas No:253585-17-0

R&D Labs maybe for 253585-17-0

Zibo Kunran Enterprises Co. LTD

website:http://www.kunranchem.com

Contact:0086 533 5200669

Address:No. 96 Jinjing Avenue, Zibo, Shandong, China
Shanghai Rechem Science Co., Ltd.

website:http://www.rechemscience.com/

Contact:+86-21-51623867

Address:Shanghai
Wuhan Yitongtai Science and Technology Co.,Ltd.

Contact:+86-27-88933550

Address:27th Fl. Bldg. 1, Shuian International Mansion, Heping Ave, Wuhan, Hubei, China
Zhangjiagang Golden Reach Fine Chemical Co.,LTD.

Contact:+86-512-6585 6968

Address:Changfu Road， Dongsha Chemical Industry Park, Zhangjiagang City, Jiangsu Province, China
taicang liyuan chemical co,.ltd

website:http://www.tcliyuanchem.com/productse.php

Contact:86-512-53539583

Address:Room 804,Huaxu Building,No.95,Renmin South Road,Taicang city,Jiangsu Province,China

Relevant to this article

Metal-free arylation of oxygen nucleophiles with diaryliodonium salts

Doi:10.1002/chem.201201645
(2012)
Gold(I)-catalyzed intramolecular amination of allylic alcohols with alkylamines

Doi:10.1021/ol103175w
(2011)
Design, synthesis and evaluation of novel tacrine-multialkoxybenzene hybrids as dual inhibitors for cholinesterases and amyloid beta aggregation

Doi:10.1016/j.bmc.2010.12.022
(2011)
Preparation and evaluation of trisubstituted pyrimidines as phosphatidylinositol 3-kinase inhibitors. 3-Hydroxyphenol analogues and bioisosteric replacements

Doi:10.1016/j.bmc.2010.12.006
(2011)
[2,2']paracyclophane-based π -conjugated molecular wires reveal molecular-junction behavior

Doi:10.1021/ja109745a
(2011)
Boosting the Catalytic Performance of Organic Salts for the Fast and Selective Synthesis of α-Alkylidene Cyclic Carbonates from Carbon Dioxide and Propargylic Alcohols

Doi:10.1002/cctc.201800063
(2018)

Article Doi