A new approach to the synthesis of efaroxan

DOI: 10.1016/S0960-894X(99)00530-2

Source and publish data:

Bioorganic and Medicinal Chemistry Letters p. 3023 - 3026 (1999)

Update date:2022-07-31

Topics:

Authors:

Couture Couture

Gouverneur

Mioskowski

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1016/S0960-894X(99)00530-2

Efaroxan was synthetised by cyclisation of the tertiary alcohol 2 which was prepared by the ring opening of the gem-disubstituted epoxide 3 with ortho-metallated fluorobenzene.

Full text of DOI:10.1016/S0960-894X(99)00530-2

Products guided by the article

Product name:2-benzyloxymethyl-2-ethyl-2,3-dihydro-benzofuran

Cas No:253585-17-0

R&D Labs maybe for 253585-17-0

shanghai payne pharm co.,ltd.

Contact:+86-021-58123769

Address:No.780 of Cailun Road,Zhangjiang Hi-tech Park,Pudong,Shanghai
Ningbo J&S Botanics Inc.

Contact:86-574-26865651

Address:529 YuanBaoShan Road, Beilun District
Zhejiang Hoshine Silicon Industry Co., Ltd.

Contact:86-573-89179966

Address:Zhapu Town, Pinghu City, Zhejiang, China
SHIFANG SUHONG CHEMICAL CO.,LTD

Contact:+86-838-2224563

Address:Room 1207 Zongchen Sunshine No.128 Taishan South Road,Deyang City,Sichuan China
sichuan tiancai fine co LTD.

website:http://www.tcfinechem.com/

Contact:18681346930

Address:baifu town,whou district

Relevant to this article

Metal-free arylation of oxygen nucleophiles with diaryliodonium salts

Doi:10.1002/chem.201201645
(2012)
Gold(I)-catalyzed intramolecular amination of allylic alcohols with alkylamines

Doi:10.1021/ol103175w
(2011)
Design, synthesis and evaluation of novel tacrine-multialkoxybenzene hybrids as dual inhibitors for cholinesterases and amyloid beta aggregation

Doi:10.1016/j.bmc.2010.12.022
(2011)
Preparation and evaluation of trisubstituted pyrimidines as phosphatidylinositol 3-kinase inhibitors. 3-Hydroxyphenol analogues and bioisosteric replacements

Doi:10.1016/j.bmc.2010.12.006
(2011)
[2,2']paracyclophane-based π -conjugated molecular wires reveal molecular-junction behavior

Doi:10.1021/ja109745a
(2011)
Boosting the Catalytic Performance of Organic Salts for the Fast and Selective Synthesis of α-Alkylidene Cyclic Carbonates from Carbon Dioxide and Propargylic Alcohols

Doi:10.1002/cctc.201800063
(2018)

Article Doi