Asymmetric synthesis of aziridinyl phosphonates using Darzens-type reaction of chloromethyl phosphonate to chiral sulfinimines

DOI: 10.1080/00397910008087297

Source and publish data:

Synthetic Communications p. 87 - 95 (2000)

Update date:2022-08-03

Topics:

Authors:

Kim, Dae Young

Suh, Ki Hyung

Choi, Jin Seok

Mang, Joo Yang

Chang, Sung Keun

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Article abstract of DOI:10.1080/00397910008087297

Darzens-type reaction of chloromethyl phosphonate with (S)-(+)-N- sulfinimines gave (Ss, 2S, 3R)-diethyl 3-aryl-2-N-(p- toluenesulfinyl)aziridinylphosphonate (3) in good yields.

Full text of DOI:10.1080/00397910008087297

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Product name:Phosphonic acid, [(2S,3R)-1-[(4-methylphenyl)sulfonyl]-3-phenyl-2-aziridinyl]-, diethyl ester

Cas No:260980-56-1

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