Bioorganic Chemistry (2019)
Update date:2022-09-26
Topics:
Chamduang, Chanamon
Pingaew, Ratchanok
Prachayasittikul, Veda
Prachayasittikul, Supaluk
Ruchirawat, Somsak
Prachayasittikul, Virapong
Novel thirteen triazole-tetrahydroisoquinoline derivatives (2a-m) were synthesized and evaluated for their aromatase inhibitory activities. Seven triazoles showed significant aromatase inhibitory activity (IC50 = 0.07–1.9 μM). Interestingly, th
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