Improved delivery through biological membranes. 32. Synthesis and biological activity of brain-targeted delivery systems for various estradiol derivatives

DOI: 10.1021/jm00396a038

Source and publish data:

Journal of Medicinal Chemistry p. 244 - 249 (1988)

Update date:2022-08-02

Topics:

Authors:

Brewster

Estes Estes

Bodor Bodor

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Article abstract of DOI:10.1021/jm00396a038

Brain-targeted delivery systems based on the dihydropyridine ? pyridinium salt redox interconversion were synthesized for estradiol, estradiol 3-benzoate, and ethynylestradiol. Initial biological evaluation indicated that while all four compounds synthesi

Full text of DOI:10.1021/jm00396a038

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