Improved delivery through biological membranes. 32. Synthesis and biological activity of brain-targeted delivery systems for various estradiol derivatives

DOI: 10.1021/jm00396a038

Source and publish data:

Journal of Medicinal Chemistry p. 244 - 249 (1988)

Update date:2022-08-02

Topics:

Authors:

Brewster

Estes Estes

Bodor Bodor

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1021/jm00396a038

Brain-targeted delivery systems based on the dihydropyridine ? pyridinium salt redox interconversion were synthesized for estradiol, estradiol 3-benzoate, and ethynylestradiol. Initial biological evaluation indicated that while all four compounds synthesi

Full text of DOI:10.1021/jm00396a038

Products guided by the article

Product name:3-<(phenylcarbonyl)oxy>-17β-<(3-pyridinylcarbonyl)oxy>estra-1,3,5(10)-triene

Cas No:4263-55-2

R&D Labs maybe for 4263-55-2

Changde Yungang Biotechnology Co., Ltd

website:http://www.cdyg.com

Contact:+86-736-7391178

Address:Qiaonan Industrial Park, Changde City, Hunan Province
Wuxi Forest Biological Co.,Ltd

Contact:+86-510-81602300

Address:Room 317,Building D, No.159 middle Chengjiang Road,Jiangyin Wuxi city.
ZHEJIANG SYNOSE TECH CO.,LTD.

website:https://www.synose.com/

Contact:86-579-82275537

Address:No.1958 Liyu Road , jinhua,zhejiang,China
HuiFeiChem PharmaTech Co.Ltd

Contact:0510-85393305

Address:1619 Huishan Avenue, Huishan District, Wuxi,
shijiazhuang alkay chemicals co..ltd(expird)

Contact:86-311-67692035

Address:2601,juntang building,qiaodong district,shijiazhuang

Relevant to this article

Synthesis, characterization, and cytotoxicity of platinum(II)/palladium(II) complexes with 4-toluenesulfonyl-L-amino acid dianion and diimine/diamine

Doi:10.1080/00958972.2013.767447
(2013)
Synthesis and properties of oligonucleotides containing 5-aza-2′-deoxycytidine

Doi:10.1080/07328319708006144
(1997)
5-Imidazolyl-quinolinones, -quinazolinones and -benzo-azepinones as farnesyltransferase inhibitors

Doi:10.1016/S0960-894X(03)00180-X
(2003)
Synthesis and molecular modeling of new 1-aryl-3-[4-arylpiperazin-1-yl]-1-propane derivatives with high affinity at the serotonin transporter and at 5-HT_1A receptors

Doi:10.1021/jm0111200
(2002)
Doi:10.1021/jm00314a008
(1967)
Synthesis, structure, and reactivity of mixed-metal clusters bearing η¹-acetylide groups, (η⁵-C₅H₅)MFe₂(μ₃-E )₂(CO)₆(η¹-CCPh) (M = Mo or W and E = Se or Te)

Doi:10.1021/om020064d
(2002)

Article Doi