Bioorganic Chemistry p. 699 - 713 (2019)
Update date:2022-08-15
Topics:
Ge, Weizhi
Liu, Zhongquan
Sun, Yu
Wang, Tianpeng
Guo, Hongyu
Chen, Xinyi
Li, Shengzu
Wang, Mengmeng
Chen, Yue
Ding, Yahui
Zhang, Quan
A series of parthenolide-SAHA hybrids were synthesized and evaluated for their anti-AML activities against HL-60 and HL-60/ADR cell lines. The most active compound 26 exhibited high activity against HL-60/ADR cell line with IC50 value of 0.15 μ
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Doi:10.1016/S0022-1139(00)80888-X
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