N-methyl as a bioisostere for the oxygen link between the aromatic rings of aryloxyphenoxypropionate herbicides

DOI: 10.1016/S0960-894X(97)00235-7

Source and publish data:

Bioorganic and Medicinal Chemistry Letters p. 1489 - 1492 (1997)

Update date:2022-08-05

Topics:

Authors:

Bird, Graham J.

Cross, Lindsay E.

Farquharson, Graeme J.

Jensen, Wendy A.

Lydiate, Jack

Serban, Alexander

Warner, Richard B.

Watson, Keith G.

Barton, John E. D.

Coles, Chris

Collins, David J.

Slater, John W.

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Article abstract of DOI:10.1016/S0960-894X(97)00235-7

The herbicidal activity of a set of N-methyl arylaminophenoxypropionate esters 3 has been compared to the analogous aryloxyphenoxypropionates 1. The usefulness of N-methyl as a novel bioisostere for ether links is shown by the surprisingly high herbicidal activity of the 6-chloroquinazolin-2-yl- and 7-chloro-1,2,4-benzotriazin-3-yl-N-methylamino- phenoxypropionate esters 3h and 3i.

Full text of DOI:10.1016/S0960-894X(97)00235-7

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