SYNTHESIS OF OPTICALLY PURE ENKEPHALIN ANALOG, ENKEPHALIN, USING CHIRAL β-LACTAMS AS SYNTHETIC INTERMEDIATES

DOI: 10.1246/cl.1982.445

Source and publish data:

Chemistry Letters p. 445 - 448 (1982)

Update date:2022-08-04

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Authors:

Hatanaka, Naoto

Abe, Rumiko

Ojima, Iwao

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Article abstract of DOI:10.1246/cl.1982.445

Optically pure pentapeptide, L-Tyr-D-Ala-Gly-L-Phe-L-Leu-ol (1) wich is an analog of opioid hormone. enkephalin, was succesfully synthesized by using β-lactam building blocks as synthons of peptide units.

Full text of DOI:10.1246/cl.1982.445

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