
Journal of Medicinal Chemistry p. 1488 - 1492 (1982)
Update date:2022-07-29
Topics: Chelation Radiolabeling Biodistribution Radiochemical purity Half-life (t?) Estrogen Receptor (ER)
Sadek
Kessler
Shaw
Anderson
Wolf
A series of seven D ring substituted selenium derivatives of estrone/estradiol has been prepared and characterized. Competitive binding studies using the rat uterine cytosol assay are reported for each compound. The most promising agent currently appears
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