Racemisation-free Esterification of 2-Nitrophenylsulphenyl-protected Amino-acids by Dicyclohexylcarbodi-imide-4-Dimethylaminopyridine

DOI: 10.1039/c39820001132

Source and publish data:

Journal of the Chemical Society. Chemical communications p. 1132 - 1133 (1982)

Update date:2022-08-04

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Authors:

Neises, Bernhard

Andries, Thomas

Steglich, Wolfgang

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Article abstract of DOI:10.1039/c39820001132

Racemisation during esterification of N-protected amino-acids by dicyclohexylcarbodi-imide-4-dimethylaminopyridine (DDC-DMAP) can be avoided by use of the 2-nitrophenylsulphenyl (Nps) protecting group.

Full text of DOI:10.1039/c39820001132

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