Tetrahedron Letters p. 983 - 985 (2019)
Update date:2022-08-04
Topics:
Wang, Xiao
Ahn, Jung-Eun
Fiejtek, Dawid K.
Lin, Lin
Dinkelborg, Katja
Sundaram, Ravi
Zheng, Shao-Liang
Iliopoulos, Othon
Hodgetts, Kevin J.
The Iliopoulos laboratory previously reported the discovery of compound 76, a small molecule HIF2α inhibitor. HIF2α activation is known to play a critical role in both von Hippel-Lindau (VHL) disease-related tumors and sporadic renal cell carcinoma (RCC).
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