Bioorganic and Medicinal Chemistry Letters p. 2721 - 2724 (2011)
Update date:2022-09-26
Topics:
Imbriglio, Jason E.
Dirocco, Daniel
Bodner, Rena
Raghavan, Subharekha
Chen, Weichun
Marley, Daria
Esser, Craig
Holt, Tom G.
Wolff, Michael S.
Taggart, Andrew K.P.
Waters, M. Gerard
Tata, James R.
Colletti, Steven L.
Amino-anthranilic acid derivatives have been identified as a new class of low serum shifted, high affinity full agonists of the human orphan G-protein-coupled receptor GPR109a with improved ADME properties.
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