Sulfur-interrupted 8-amino side chain analogues of 4-methyl-5-[m-(trifluoromethyl)phenoxy]primaquine as potential antimalarial agents

DOI: 10.1021/jm00150a035

Source and publish data:

Journal of Medicinal Chemistry p. 1959 - 1962 (1985)

Update date:2022-08-04

Topics:

Authors:

Carroll Carroll

Berrang Berrang

Linn Linn

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Article abstract of DOI:10.1021/jm00150a035

Two isomeric sulfur-interrupted 8-amino side chain analogues of 4-methyl-5-[m-(trifluoromethyl)phenoxy]primaquine (2) were prepared and tested for antimalarial activity. The compounds were evaluated for blood schizonticidal activity aginst Plasmodium berg

Full text of DOI:10.1021/jm00150a035

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