An efficient synthesis of 2-(((9- fluorenylmethoxycarbonyl)amino)methyl)benzoic acid

Article abstract of DOI:10.1080/00397919808004516

An efficient, two-step synthesis of the title compound 3 in 61% overall yield is presented. The synthesis involves hydrazine removal of the N- phthalimide protecting group of α-phthalimido-o-toluic acid (6), followed by N-Fmoc formation with (9-fluorenylm

Full text of DOI:10.1080/00397919808004516

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An Efficient
Synthesis of 2-(((9-
Fluorenylmethoxycarbonyl)amin
Acid
a
a
Jung-Hui Sun & Wayne F. Daneker
a
The DuPont Merck Pharmaceutical Company ,
Experimental Station , P.O. Box 80336,
Wilmington, DE, 19880-0336
Published online: 22 Aug 2006.
To cite this article: Jung-Hui Sun & Wayne F. Daneker (1998) An Efficient
Synthesis of 2-(((9-Fluorenylmethoxycarbonyl)amino)methyl)benzoic Acid,
Synthetic Communications: An International Journal for Rapid Communication of
Synthetic Organic Chemistry, 28:24, 4525-4530, DOI: 10.1080/00397919808004516
To link to this article: http://dx.doi.org/10.1080/00397919808004516
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