18F-labelling of a potent nonpeptide CCR1 antagonist: Synthesis of 1-(5-chloro-2-{2-[(2r)-4-(4-[18F]fluorobenzyl)-2-methylpiperazin- 1-yl]-2-oxoethoxy}phenyl)urea in an automated module

DOI: 10.1002/jlcr.1023

Source and publish data:

Journal of labelled compounds and radiopharmaceuticals p. 253 - 262 (2006)

Update date:2022-08-10

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Authors:

Maeding Maeding

Fuechtner

Johannsen

Steinbach

Hilger Hilger

Friebe Friebe

Halks-Miller

Horuk Horuk

Mohan Mohan

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Article abstract of DOI:10.1002/jlcr.1023

The synthesis of 1-(5-chloro-2-{2-[(2R)-4-(4-[¹⁸F]fluorobenzyl)- 2-methylpiperazin-1-yl]-2-oxoethoxy}phenyl)urea ([¹⁸F]4), a potent nonpeptide CCR1 antagonist, is described as a module-assisted two-step one-pot procedure. The final p

Full text of DOI:10.1002/jlcr.1023

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