Chemistry - An Asian Journal p. 1832 - 1838 (2021)
Update date:2022-07-29
Topics:
Zhang, Qinglin
Duan, Yongbin
Guo, Huifeng
Yang, Hong
Zhai, Jiulong
Li, Tiantian
Wang, Zhihai
Lu, Xiaolei
Wang, Yan
Yin, Yan
A Bi(OTf)3-catalyed reaction of 3-aryl propargyl alcohols with sulfonamide and halogen source was firstly investigated, which provided a facile route for the synthesis of a large variety of α-halo-β-amino ketones. The key intermediates, β-amino
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