Synthesis and Benzodiazepine Binding Activity of a Series of Novel Triazoloquinazolin-5(6H)-ones

DOI: 10.1021/jm00105a044

Source and publish data:

Journal of Medicinal Chemistry p. 281 - 290 (1991)

Update date:2022-08-04

Topics:

Authors:

Francis, John E.

Cash, William D.

Barbaz, Beverly S.

Bernard, Patrick S.

Lovell, Richard A.

et al. et al.

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Article abstract of DOI:10.1021/jm00105a044

Investigation of tricyclic heterocycles related to the 2-arylpyrazolo<4,3-c>quinolin-3(5H)-ones, structures with high affinity for the benzodiazepine (BZ) receptor, led to the synthesis of 2-phenyl-<1,2,4>triazolo<1,5-c>quinazolin-5(6H)-one, a compound wi

Full text of DOI:10.1021/jm00105a044

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