Bioorganic and Medicinal Chemistry Letters p. 3279 - 3282 (2009)
Update date:2022-08-04
Topics:
Mizuguchi, Takaaki
Uchimura, Hiromasa
Kakizawa, Taeko
Kimura, Tooru
Yokoyama, Shigeyuki
Kiso, Yoshiaki
Saito, Kazuki
A cyclic decapeptide was chemically synthesized that mimics the loop structure of a β-hairpin arm of the EGF receptor, which is highly involved in receptor dimerization upon activation by ligand binding. This peptide was revealed to reduce dimer formation
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