Probes for Narcotic Receptor Mediated Phenomena. 15. (3S,4S)-(+)-trans-3-Methylfentanyl Isothiocyanate, a Potent Site-Directed Acylating Agent for the δ Opioid Receptors in Vitro

DOI: 10.1021/jm00126a040

Source and publish data:

Journal of Medicinal Chemistry p. 1392 - 1398 (1989)

Update date:2022-08-02

Topics:

Authors:

Kim, Chong-Ho

Rothman, Richard B.

Jacobson, Arthur E.

Mattson, Mariena V.

Bykov, Victor

et al. et al.

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1021/jm00126a040

Recently we reported the synthesis of the first enantiomeric pair of irreversible opioid ligands <(3S,4R)-(-)- and (3R,4S-(+)-cis-4, SUPERFIT> and specific interaction of the latter with the δ receptor.Here we report another enantiomeric pair of irreversi

Full text of DOI:10.1021/jm00126a040

Products guided by the article

Product name:(3R,4R)-trans-N-<1-<2-(4-Isothiocyanatophenyl)ethyl>-3-methyl-4-piperidyl>-N-phenylpropanamide

Cas No:120143-77-3

R&D Labs maybe for 120143-77-3

Zhejiang Kangfeng Chemical Co.,LTD.

Contact:+86-579-86709687

Address:Xueshizhai Industrial Zone, Weishan Town,Dongyang City, Zhejiang Province ,China
Shanghai Surseechem Co.,Ltd.

Contact:+86-21-61318535

Address:Building 29,No.2139 Xizha Road, Fengxian District, Shanghai
Tianjin Jiuri New Materials Co., Ltd.

Contact:+86-22-58889220

Address:C-5/6, Vison Hill, No.1 Gonghua Road, Huayuan Hi-tech Park, Tianjin, China.
TIANJIN DONGRUXIANG MINERALS MARKETING CO.,LTD(expird)

Contact:22-58516360

Address:tianjin
Buffett (China) Holding Co.,Ltd

Contact:4006570891

Address:

Relevant to this article

THE CHEMISTRY OF PENTAVALENT ORGANOBISMUTH REAGENTS. PART XI. REACTIONS WITH STERICALLY HINDERED PHENOLS.

Doi:10.1016/S0040-4020(01)86150-0
(1988)
SYNTHESIS OF α,α-DICHLORO-β-HYDROXYNITRILE MEDIATED BY TRI-n-BUTYLSTIBINE

Doi:10.1016/S0040-4039(00)80735-2
(1988)
Solution to the C₃-Arylation of Indazoles: Development of a Scalable Method

Doi:10.1021/acs.orglett.6b01456
(2016)
Evaluation of adenine as scaffold for the development of novel P2X3 receptor antagonists

Doi:10.1016/j.ejmech.2013.04.037
(2013)
Synthesis of α-aminonitriles through Strecker reaction of N-tosylaldimines using molecular iodine

Doi:10.1055/s-0029-1216969
(2009)
Synthesis, crystal structure and biological activity of N′-tert-butyl-N-(3-methoxylbenzoyl)-N-(4-methyl-1,2, 3-thiadiazole-5- formylhydrazine

Doi:10.1007/s10870-011-0189-1
(2011)

Article Doi