ONE POT SYNTHESIS OF HOMOCHIRAL AZIRIDINES AND AMINOALCOHOLS FROM HOMOCHIRAL 1,2-CYCLIC SULFATES

Article abstract of DOI:10.1016/S0040-4039(00)99081-6

Preparations of homochiral N-substituted aziridines and aminoalcohols from 1,2-cyclic sulfates are reported.Primary amines react with cyclic sulfates to give β-aminosulfates which can be converted either to aziridines or to aminoalcohols by treatment with