MITSUNOBU REACTIONS OF N-ALKYL AND N-ACYL SULFONAMIDES - AN EFFICIENT ROUTE TO PROTECTED AMINES

DOI: 10.1016/S0040-4039(00)76177-6

Source and publish data:

Tetrahedron Letters p. 5709 - 5712 (1989)

Update date:2022-09-26

Topics: Mitsunobu reactions N-alkyl sulfonamides

Authors:

Henry, James R.

Marcin, Lawrence R.

McIntosh, Matthias C.

Scola, Paul M.

Harris, G. Davis

Weinreb, Steven M.

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Article abstract of DOI:10.1016/S0040-4039(00)76177-6

N-Methyl p-toluenesulfonamide and N-BOC p-toluenesulfonamide can be directly coupled with primary or secundary alcohols under Mitsunobu conditions to afford various sulfonamide-protected amines.

Full text of DOI:10.1016/S0040-4039(00)76177-6

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