Asymmetric Synthesis of α-Alkylated Tryptophan Derivatives

DOI: 10.1039/c39890001418

Source and publish data:

Journal of the Chemical Society. Chemical communications p. 1418 - 1419 (1989)

Update date:2022-08-03

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Authors:

Crich, David

Davies, John W.

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Article abstract of DOI:10.1039/c39890001418

L-Tryptophan has been converted, by the alkylation of the hexahydro<2,3-b>pyrropoindole (7), followed by ring opening, to α-alkylated tryptophan derivatives with overall retention of configuration.

Full text of DOI:10.1039/c39890001418

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