Modification of the Enkephalin "Message" with an Artificial Polycationic C-Terminus

DOI: 10.1021/jm00113a020

Source and publish data:

Journal of Medicinal Chemistry p. 2816 - 2821 (1991)

Update date:2022-09-26

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Authors:

Jacobson, Alan R.

Tam, S. William

Sayre, Lawrence M.

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Article abstract of DOI:10.1021/jm00113a020

The C-terminal "address" sequences of prodynorphin-derived opioid peptides contain an unusually high proportion of basic residues, which are known to be crucial for conferring high activity and selectivity for κ-opioid receptors.In an effort to investigat

Full text of DOI:10.1021/jm00113a020

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