Structure-Antigastrin Activity Relationships of New (R)-4-Benzamido-5-oxopentanoic Acid Derivatives

DOI: 10.1021/jm00079a003

Source and publish data:

Journal of Medicinal Chemistry p. 28 - 38 (1992)

Update date:2022-09-26

Topics:

Authors:

Makovec, Francesco

Peris, Walter

Revel, Laura

Giovanetti, Roberto

Mennuni, Laura

Rovati, Lucio C.

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Article abstract of DOI:10.1021/jm00079a003

New (R)-4-benzamido-5-oxopentanoic acid derivatives were synthesized by a stereoconservative procedure and evaluated in vitro for their capacity to inhibit the binding of <125I>(BH)-CCK-8 to either rat peripheral (CCK-A) or central (CCK-B) CCK receptors,

Full text of DOI:10.1021/jm00079a003

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Product name:(R)-4-Benzyloxycarbonylamino-5-(4,4-dimethyl-piperidin-1-yl)-5-oxo-pentanoic acid benzyl ester

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