Structure-Antigastrin Activity Relationships of New (R)-4-Benzamido-5-oxopentanoic Acid Derivatives

DOI: 10.1021/jm00079a003

Source and publish data:

Journal of Medicinal Chemistry p. 28 - 38 (1992)

Update date:2022-09-26

Topics:

Authors:

Makovec, Francesco

Peris, Walter

Revel, Laura

Giovanetti, Roberto

Mennuni, Laura

Rovati, Lucio C.

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1021/jm00079a003

New (R)-4-benzamido-5-oxopentanoic acid derivatives were synthesized by a stereoconservative procedure and evaluated in vitro for their capacity to inhibit the binding of <125I>(BH)-CCK-8 to either rat peripheral (CCK-A) or central (CCK-B) CCK receptors,

Full text of DOI:10.1021/jm00079a003

Products guided by the article

Product name:(R)-4-Benzyloxycarbonylamino-5-(4,4-dimethyl-piperidin-1-yl)-5-oxo-pentanoic acid benzyl ester

Cas No:137795-79-0

R&D Labs maybe for 137795-79-0

Rizhao Lanxing Chemical Indusrial Co.,Ltd

Contact:86-633-2616708

Address:NO.15 West road Shenglan, Lanshan district, Rizhao City
Zhejiang Hoshine Silicon Industry Co., Ltd.

Contact:86-573-89179966

Address:Zhapu Town, Pinghu City, Zhejiang, China
HANGZHOU FOREWIN PHARMA CO., LTD

Contact:+86-571-89053961

Address:hangzhou
Shanghai Rich Chemicals Co., Ltd

website:http://www.richchemical.com

Contact:+86-21-20255798

Address:Pudong Shanghai,China
Chengdu Herbpurify Co., Ltd

website:http://www.herbpurify.com

Contact:0086-028-85249238

Address:Room709-C1,Incubator Building, Tianfu Life Science Park No.88,Keyuan Road,Gaoxin district,Chengdu City,Sichuan Prov,China

Relevant to this article

ASYMMETRIC SYNTHESIS OF TOPOGRAPHICALLY CONSTRAINED AMINO ACIDS: SYNTHESIS OF THE OPTICALLY PURE ISOMERS OF α,β-DIMETHYL-PHENYLALANINE AND α,β-DIMETHYL-1,2,3,4-TETRAHYDROISOQUINOLINE-3-CARBOXYLIC ACID

Doi:10.1016/S0040-4039(00)93551-2
(1991)
Synthesis of halogenated α,β-unsaturated γ-butyrolactone derivatives by triphenylphosphine-catalyzed cyclization of α-halogeno ketones with dialkyl acetylenedicarboxylates (=dialkyl but-2-ynedioates)

Doi:10.1002/hlca.201100376
(2012)
KO^tBu mediated synthesis of phenanthridinones and dibenzoazepinones

Doi:10.1021/ol301077y
(2012)
Facile and convenient synthesis of functionalized aryl-containing isoindigo derivatives via substituted indolin-2-one carbene dimerization

Doi:10.1080/00397911.2011.558232
(2012)
Carbenylative amination with N-tosylhydrazones

Doi:10.1021/ol301385g
(2012)
Doi:10.1021/jo01349a020
(1966)

Article Doi