Preparation of Chiral Aziridines from Chiral Oxiranes with Retention of Configuration

DOI: 10.1039/c39920000284

Source and publish data:

Journal of the Chemical Society. Chemical communications p. 284 - 285 (1992)

Update date:2022-08-04

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Authors:

Toshimitsu, Akio

Abe, Hideyuki

Hirosawa, Chitaru

Tanimoto, Shigeo

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Article abstract of DOI:10.1039/c39920000284

Chiral oxiranes are converted into chiral aziridines via β-hydroxyalkyl aryl sulfides and then β-tosylaminoalkyl aryl sulfides without loss of optical purity and with overall retention of configuration.

Full text of DOI:10.1039/c39920000284

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