Design, synthesis, and pharmacology of 3-substituted sodium azulene-1- sulfonates and related compounds: Non-prostanoid thromboxane A2 receptor antagonists

DOI: 10.1021/jm00059a001

Source and publish data:

Journal of Medicinal Chemistry p. 791 - 800 (1993)

Update date:2022-08-05

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Authors:

Tomiyama

Yokota Yokota

Wakabayashi

Kosakai Kosakai

Yanagisawa

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Article abstract of DOI:10.1021/jm00059a001

A series of novel azulene-1 carboxylic acid derivatives 28-30, azulene-1 sulfonic acid sodium salts 41a-c, and related compounds were synthesized. These compounds were tested for TXA₂ receptor antagonistic activity. The inhibitory concentration

Full text of DOI:10.1021/jm00059a001

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Product name:methyl 3-<3-<(benzyloxy)methyl>phenyl>-6-isopropylazulene-1-carboxylate

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