Tetrahedron Letters p. 3483 - 3486 (1997)
Update date:2022-08-04
Topics:
Branalt, Jonas
Kvarnstroem, Ingemar
Classon, Bjoern
Samuelsson, Bertil
Nillroth, Ulrika
Danielson, U. Helena
Karlen, Anders
Hallberg, Anders
A new short route to epoxide 6b, a pivotal intermediate for the preparation of hydroxyethylamine dipeptide isosteres has been developed. Opening of the epoxide by anthranilic acid, followed by extensions in the P2/P3-region gave the target compounds which were evaluated as HIV-1 protease inhibitors.
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