Stereoselective Synthesis of trans-2-(Indol-3-yl)cyclopropylamines: Rigid Tryptamine Analogues

DOI: 10.1021/jo00116a028

Source and publish data:

Journal of Organic Chemistry p. 3409 - 3413 (1995)

Update date:2022-08-04

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Authors:

Vangveravong, Suwanna

Nichols, David E.

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Article abstract of DOI:10.1021/jo00116a028

A procedure for the preparation of trans-2-(indol-3-yl)cyclopropylamines is reported.The key step in the sequence is a stereoselective palladium-catalyzed cyclopropanation of the indole-3-acryloyl derivative of Oppolzer's chiral sultam (bornane<10,2>sulta

Full text of DOI:10.1021/jo00116a028

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Product name:trans-β-<1-(p-Toluenesulfonyl)indol-3-yl>acryloyl chloride

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